680860-46-2

Upstream product

• 680860-37-1 N-allyl-5-fluoro-2-nitro-N-(1-phenyl-ethyl)-benzamide 
• 680860-40-6 N-allyl-2-amino-5-fluoro-N-(1-phenyl-ethyl)-benzamide 
• 680860-35-9 5-fluoro-2-nitro-N-(1-phenyl-ethyl)-benzamide 
• 3886-69-9 (R)-1-phenyl-ethyl-amine 
• 394-02-5 5-fluoro-2-nitrobenzoyl chloride 
• 680860-43-9 N-allyl-2-azido-5-fluoro-N-(1-phenyl-ethyl)-benzamide 

Relevant academic research and scientific papers

Diastereoselective synthesis of enantiopure (αR)-2-methyl-4-(α- phenylethyl)-1,2,3,4-tetrahydro-benzo[e][1,4]diazepin-5-ones

(αR,2R)- and (αR,2S)-2-methyl-4-(α-phenylethyl)-1,2,3,4- tetrahydro-benzo[e][1,4]diazepin-5-ones 7 and 8 were synthesised by an intramolecular azide cycloaddition followed by stereoselective reduction of a bicyclic ketimine.