697304-21-5Relevant articles and documents
A practical synthesis of enantiopure β-methyltryptophan ethyl ester for a preparation of diabetes drug
Sawai, Yasuhiro,Mizuno, Masahiro,Ito, Tatsuya,Kawakami, Jun-ichi,Yamano, Mitsuhisa
experimental part, p. 7122 - 7128 (2009/12/06)
A practical synthesis of (2R,3S)- and (2S,3R)-β-methyltryptophan ethyl ester (β-MeTrp-OEt) has been developed. Racemic threo-β-MeTrp-OEt was diastereoselectively prepared via crystallization-induced diastereomer transformation (CIDT) of the α-nitro equiva