714567-80-3Relevant articles and documents
Development of an efficient and selective radioligand for bradykinin B 1 receptor occupancy studies
Su, Dai-Shi,Markowitz, M. Kristine,Murphy, Kathy L.,Wan, Bang-Lin,Zrada, Matthew M.,Harrell, C. Meacham,O'Malley, Stacy S.,Hess, J. Fred,Ransom, Rick W.,Chang, Ray S.,Wallace, Michael A.,Raab, Conrad E.,Dean, Dennis C.,Pettibone, Douglas J.,Freidinger, Roger M.,Bock, Mark G.
, p. 6045 - 6048 (2004)
We have developed an efficient and selective radioligand, the [ 35S]-radiolabeled dihydroquinoxalinone derivative, 4, for an ex vivo receptor occupancy assay in transgenic rats over-expressing the human bradykinin B1 receptor.