749912-25-2Relevant academic research and scientific papers
Solution-phase parallel synthesis and evaluation of anticonvulsant activity of N-substituted-3,4-dihydroisoquinoline-2(1H)-carboxamides
Gitto, Rosaria,Pagano, Benedetta,Citraro, Rita,Scicchitano, Francesca,De Sarro, Giovanbattista,Chimirri, Alba
experimental part, p. 1349 - 1354 (2009/09/27)
In our previous studies we identified several isoquinoline derivatives displaying potent anticonvulsant effects in different animal models of epilepsy. With the aim to exploit the main structure-activity relationships (SAR) for this class of compounds we
