75371-60-7Relevant academic research and scientific papers
A metal-free multicomponent cascade reaction for the regiospecific synthesis of 1,5-disubstituted 1,2,3-triazoles
Cheng, Guolin,Zeng, Xiaobao,Shen, Jinhai,Wang, Xuesong,Cui, Xiuling
supporting information, p. 13265 - 13268 (2014/01/06)
About specifics: A method for the regiospecific synthesis of the title compounds through an unprecedented Michael addition/deacylative diazo transfer/cyclization sequence has been established. The simple and practical method can be used for the modification of primary amines including chiral α-amines. The process involves the formation three covalent bonds and the cleavage of two covalent bonds (see scheme, Ts=4-toluenesulfonyl).
Reactions of Primary and Secondary Aromatic Amines with Aroylphenylacetylenes and Configurational Assignments of the Adducts
Fouli, F. A.,Beshay, A. D.
, p. 410 - 412 (2007/10/02)
The reaction of aroylphenylacetylenes (Ia-c) with aniline and other primary and secondary aromatic amines in a protic solvent (ethanol) gives rise to only (Z)-isomers (IIa-s) of the adducts.However, the reaction of benzoylphenylacetylene (Ia) with aniline
