75371-68-5Relevant academic research and scientific papers
Copper-promoted Chan-Lam coupling between enaminones and aryl boronic acids
Duan, Xiyan,Liu, Ning,Liu, Kun,Song, Yakun,Wang, Jia,Mao, Xianhua,Xu, Weidong,Yang, Shijie,Li, Huixian,Ma, Junying
supporting information, p. 4187 - 4190 (2018/10/24)
A novel copper-promoted N-arylation of enaminones with aromatic boronic acids has been developed, which provides an efficient way to synthesize N-aryl enaminones with a broad substrate scope and excellent functional group compatibility. The N-aryl enaminones could be converted into a series of highly valuable building blocks and bioactive compounds. Notably, in comparison with traditional methods, this alternative approach provides accesses to N-aryl enaminones bearing multiple aromatic rings.
Simple and efficient one-pot, three-component, solvent-free synthesis of β-enaminones via sonogashira coupling-michael addition sequences
Palimkar, Sanjay S.,More, Vijaykumar S.,Srinivasan, Kumar V.
, p. 1456 - 1469 (2008/09/21)
A simple, efficient, and environmentally friendly one-pot, three-component synthesis of β-enaminones via Sonogashira coupling-Michael addition sequences under solvent-free conditions has been reported. Also the synthesis of β-enaminones has been achieved
Synthesis and Spectral Properties of β-Anilino-α-(p-chlorobenzoyl)styrene Derivatives
Al-Hajjar, F.,Al-Sultan, Y.,Abushihada, A.,Shunbo, F.
, p. 83 - 85 (2007/10/02)
(p-Chlorobenzoyl)phenylacetylene reacted with aniline derivatives to give the corresponding β-anilino-α-(p-chlorobenzoyl)styrene derivative.NMR, UV, IR, and mass spectra of these compounds are presented.The Hammett correlation is applied to substituent ef
Reactions of Primary and Secondary Aromatic Amines with Aroylphenylacetylenes and Configurational Assignments of the Adducts
Fouli, F. A.,Beshay, A. D.
, p. 410 - 412 (2007/10/02)
The reaction of aroylphenylacetylenes (Ia-c) with aniline and other primary and secondary aromatic amines in a protic solvent (ethanol) gives rise to only (Z)-isomers (IIa-s) of the adducts.However, the reaction of benzoylphenylacetylene (Ia) with aniline
