75392-23-3Relevant articles and documents
Syntheis of 3-(1,2,3,6-tetrahydro pyridin-4-yl) 1H-indoles and study of their serotoninergic and anti-dopaminergic properties
Guillaume,Dumont,Laurent,Nedelec
, p. 33 - 43 (2007/10/02)
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Process for preparation of piperidyl-indoles
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, (2008/06/13)
A novel process for the preparation of piperidylindoles of the formula STR1 wherein R is selected from the group consisting of hydrogen and alkyl of 1 to 3 carbon atoms and X is selected from the group consisting of hydrogen, nitro, fluorine, bromine, chlorine and alkoxy of 1 to 3 carbon atoms and their non-toxic, pharmaceutically acceptable acid addition salts thereof by reacting an indole of the formula STR2 with 4-piperidone hydrochloride in an alkaline medium to obtain the compound of formula I which is optionally salified and the novel product, 5-nitro-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole and its non-toxic, pharmaceutically acceptable acid addition salts.