7564-39-8Relevant articles and documents
PYRAZOLE DERIVATIVES AS S1P1 AGONISTS
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Page/Page column 36, (2011/12/04)
The present invention relates to a compound of formula (I), to the process for preparing such compounds and to their use in the treatment of a pathological condition or disease susceptible to amelioration by sphingosine-1-phosphate receptors (S1P1) agonists.
Selected Cgrp-Antagonists, Processes for Preparing Them and Their Use as Pharmaceutical Compositions
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Page/Page column 59-60, (2008/12/08)
The invention relates to CGRP-antagonists of general formula (I), wherein R1, R2, R3, R4 and R5 are defined in claim 1, to the tautomers, isomers, diastereomers, enantiomers, hydrates, mixtures salts and salt hydrates thereof, in particular to 10 salts thereof, which are physiologically compatible with acids or inorganic or organic bases and to compounds of general formula (I), wherein one or several hydrogen atoms are substituted by deuterium. Drugs containing said compounds, the use thereof and a method for the production thereof are also disclosed.
Selected CGRP antagonists, process for their preparation as well as their use as medicaments
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, (2008/06/13)
Heterocyclic esters (I), their tautomers, diastereomers, enantiomers, hydrates, mixtures and (hydrated) salts, particularly physiologically acceptable salts with (in)organic acids and bases, that are antagonists of calcitonin gene-related peptide (CGRP) a