769126-83-2Relevant academic research and scientific papers
24,24-Dimethylvitamin D3-26,23-lactones and their 2α-functionalized analogues as highly potent VDR antagonists
Saito, Nozomi,Masuda, Manami,Matsunaga, Toshihiro,Saito, Hiroshi,Anzai, Miyuki,Takenouchi, Kazuya,Miura, Daishiro,Ishizuka, Seiichi,Takimoto-Kamimura, Midori,Kittaka, Atsushi
, p. 7951 - 7961 (2007/10/03)
Novel vitamin D receptor (VDR) antagonists, 24,24-dimethyl-1α- hydroxyvitamin D3-26,23-lactones (8 and 9) and their C2α functionalized analogues (8a-c and 9a-c) were efficiently synthesized and their biological activities were evaluated. The co
