78839-80-2Relevant articles and documents
METHODOLOGY FOR INDOLE SYNTHESIS
Wender, Paul A.,White, Alan W.
, p. 1475 - 1478 (1981)
An efficient synthesis of indole derivatives in one operation by reaction of organodilithium reagents with vicinal dication equivalents is described.
METHODOLOGY FOR THE FACILE AND REGIO-CONTROLLED SYNTHESIS OF INDOLES
Wender, Paul A.,White, Alan W.
, p. 3767 - 3776 (2007/10/02)
A method based on organodimetallic reagents is described for the regiocontrolled synthesis of indoles which proceeds, generally, in one to two operations from commercially or readily available reactants.The method is applied to the synthesis of indole itself, 2-substituted, 3-substituted, 2,3-disubstituted and 6-substituatd indoles.