78844-19-6Relevant academic research and scientific papers
Analogs of Ac-CCK-7 Incorporating Dipeptide Mimics in Place of Met28-Gly29
Tilley, Jefferson W.,Danho, Waleed,Shiuey, Shian-Jun,Kulesha, Irina,Swistok, Joseph,et al.
, p. 3774 - 3783 (2007/10/02)
A series of analogs of Ac-CCK-7 28-Gly29-Trp-Met-Asp-Phe-NH2, (1)> were prepared in which The Met28-Gly29 dipeptide was replaced by ω-aminoalkanoic acids.Compounds were assessed in binding assay
Synthesis of &γ-Aminobutyric Acid Analogue of Restricted Conformation. Part 1. The 2-Aminocycloalkylacetic Acids
Kennewell, Peter D.,Matharu, Saroop S.,Taylor, John B.,Westwood, Robert,Sammes, Peter G.
, p. 2553 - 2562 (2007/10/02)
The syntheses of cis- and trans-2-aminocyclopropyl, -cyclobutyl, -cyclopentyl, and cyclohexylacetic acids as γ-aminobutyric acid analogues of restricted conformation are described.Mass spectral evidence fully supports the stereochemical assignements of configurational isomers.
THE ASSYMETRIC MICHAEL REACTION OF (2R,3S)-3,4-DIMETHYL-2-PHENYLPERHYDRO-1,4-OXAZEPINE-5,7-DIONE WITH 1-NITROCYCLOHEXENE
Takeda, Takeshi,Hoshihiko, Tomonori,Mukaiyama, Teruaki
, p. 797 - 800 (2007/10/02)
Optically active (2-nitrocyclohexyl)acetic acid(III) was obtained by the Michael reaction of (2R,3S)-3,4-dimethyl-2-phenylperhydro-1,4-oxazepine-5,7-dione(I) with 1-nitrocyclohexene in the presence of potassium t-butoxide (or cesium fluoride) and crown et
