791809-55-7Relevant academic research and scientific papers
Design, synthesis, and biological evaluation of 4-arylmethyl-1- phenylpyrazole and 4-aryloxy-1-phenylpyrazole derivatives as novel androgen receptor antagonists
Yamamoto, Satoshi,Tomita, Naoki,Suzuki, Yuri,Suzaki, Tomohiko,Kaku, Tomohiro,Hara, Takahito,Yamaoka, Masuo,Kanzaki, Naoyuki,Hasuoka, Atsushi,Baba, Atsuo,Ito, Mitsuhiro
experimental part, p. 2338 - 2352 (2012/05/07)
A series of 4-arylmethyl-1-phenylpyrazole and 4-aryloxy-1-phenylpyrazole compounds B were designed, synthesized, and evaluated for their potential as new-generation androgen receptor (AR) antagonists therapeutically effective against castration-resistant
TRIAZINE COMPOUNDS AND THEIR USE
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Page 23, (2010/02/09)
A compound of formula (I) wherein R1 is hydrogen, alkyl, -alkyl-aryl, -alkyl-heterocycloalkyl or -alkyl-0-heterocycloalkyl; R2 is hydrogen, hydroxy, amino, nitro, alkoxy, alkyl, aryl or heteroaryl; R3 is hydrogen, alkyl or
