792912-66-4Relevant academic research and scientific papers
PHTALAZINONE DERIVATIVES AS MPEGS -1 INHIBITORS
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Page/Page column 40; 41, (2013/06/05)
The present patent application is directed to bicyclic compounds of formula (I) or pharmaceutically acceptable salt thereof as mPGES-1 inhibitors. These compounds are inhibitors of the microsomal prostaglandin E synthase-1 (m PGES-1) enzyme and are theref
BENZAMIDE INHIBITORS OF THE P2X7 RECEPTOR
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Page 95, (2008/06/13)
The present invention provides benzamide inhibitors of the P2X7 receptor of the formula (I), wherein R1 -R3 are as defined herein. The compounds of the invention are useful in the treatment of IL-1 mediated disorders, incl
