795315-07-0Relevant academic research and scientific papers
Achiral, selective CCK2 receptor antagonists based on a 1,3,5-benzotriazepine-2,4-dione template
Spencer, John,Gaffen, John,Griffin, Eric,Harper, Elaine A.,Linney, Ian D.,McDonald, Iain M.,Roberts, Sonia P.,Shaxted, Mark E.,Adatia, Trushar,Bashall, Alan
, p. 2974 - 2983 (2008/09/19)
Novel, achiral 1H-1,3,5-benzotriazepine-2,4(3H,5H)-diones have been prepared and structurally characterized. These compounds are potent CCK2 receptor antagonists that display a high degree of selectivity over CCK1 receptors.
BENZOTRIAZEPINE DERIVATIVES AND THEIR USE AS GASTRIN AND CHOLECYSTOKININ RECEPTOR LIGANDS
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Page/Page column 23, (2010/02/09)
This invention relates to a compound of formula (I). The compound is useful for the treatment of gastrin related disorders.
