795315-50-3Relevant articles and documents
Achiral, selective CCK2 receptor antagonists based on a 1,3,5-benzotriazepine-2,4-dione template
Spencer, John,Gaffen, John,Griffin, Eric,Harper, Elaine A.,Linney, Ian D.,McDonald, Iain M.,Roberts, Sonia P.,Shaxted, Mark E.,Adatia, Trushar,Bashall, Alan
, p. 2974 - 2983 (2008/09/19)
Novel, achiral 1H-1,3,5-benzotriazepine-2,4(3H,5H)-diones have been prepared and structurally characterized. These compounds are potent CCK2 receptor antagonists that display a high degree of selectivity over CCK1 receptors.