79976-76-4Relevant academic research and scientific papers
An efficient synthesis of new aza-substituted indoles via Michael-type addition
Bayindir, Sinan,Erdogan, Esra,Kilic, Haydar,Saracoglu, Nurullah
, p. 1455 - 1458 (2010)
An efficient method has been developed for the synthesis of new aza-substituted indoles. The methodology involves a two-step synthesis. The first step involves the Michael addition of indoline with various Michael acceptors. The other includes the oxidation of the indoline ring in the Michael adducts to an indole.
Synthesis of highly N-substituted indole library via conjugate additions of indoline and their synthetic tool potentials
Kilic, Haydar,Bayindir, Sinan,Erdogan, Esra,Saracoglu, Nurullah
, p. 5619 - 5630 (2012/09/08)
A comprehensive library of N- or 1-substituted indoles was formed by conjugate additions of indoline with Michael acceptors followed by an oxidation step. Using N-substituted indoles as key Michael donors, the synthesis of 1,3-disubstituted indoles was al
