80232-92-4Relevant articles and documents
SYNTHETIC APPLICATIONS OF 2-CHLOROOXIRANES: PREPARATION OF THIAZOLES, DIHYDROTHIAZOLES AND SELENAZOLES
Gasteiger, Johann,Herzig, Christian
, p. 2607 - 2611 (1981)
The reaction of 2-chlorooxiranes 1 with thioamides and thioureas provides access to thiazoles, 4-hydroxy-4,5-dihydrothiazoles and 2-imino-2,3-dihydrothiazoles under mild conditions and excellent yields.With 1 and selenourea, near quantitative yields of se
Synthesis and Mercuration of Some New 3-Aryl-2-arylimino-4,5-disubstituted-δ4-thiazolines and Their Fungicidal and Bactericidal Activities
Mohanty, J.,Mahapatra, G. N.
, p. 52 - 55 (2007/10/02)
A series of new 3-aryl-2-arylimino-4,5-disubstituted-Δ4-thiazolines (I) have been synthesised by condensing various ketones having active methylene group with sym-diarylthioureas in the presence of bromine.The thiazolines (I) on mercuration with one equivalent of mercuric acetate in acetic acid give 3-(acetoxymercuriaryl)-2-arylimino-4,5-disubstituted-Δ4-thiazolines (II).All the compounds have been assayed against the fungus Pyricularia oryzae (Cav) and the bacteria Esch. coli and Staph. aureus, and the structure-activity relationship has been discussed.