81154-09-8Relevant articles and documents
Discovery and development of novel rhodanine derivatives targeting enoyl-acyl carrier protein reductase
Xu, Jian-Fei,Wang, Tian-Tian,Yuan, Qing,Duan, Yong-Tao,Xu, Yun-Jie,Lv, Peng-Cheng,Wang, Xiao-Ming,Yang, Yu-Shun,Zhu, Hai-Liang
, p. 1509 - 1516 (2019/03/05)
A series of rhodanine derivatives RB1–RB23 were synthesized through a two-round screening. Their Mycobacterial tuberculosis (Mtb) InhA inhibitory activity and Mtb growth blocking capability were evaluated. The most potent hit compound RB23 indicated compa
Molecular docking evaluation of (E)-5-arylidene-2-thioxothiazolidin-4-one derivatives as selective bacterial adenylate kinase inhibitors
Ionescu, Mihaela Ileana,Oniga, Ovidiu
, (2018/05/22)
Multi-drug resistant microorganism infections with emerging problems that require not only a prevention strategy, but also the development of new inhibitory compounds. Six previously synthesized 5-arylidene-2-thioxothiazolidin-4-one derivatives 1a–f, were
Combination of 4-anilinoquinazoline and rhodanine as novel epidermal growth factor receptor tyrosine kinase inhibitors
Li, Si-Ning,Xu, Yun-Yun,Gao, Jia-Yu,Yin, Hong-Ran,Zhang, Shi-Lei,Li, Huan-Qiu
, p. 3221 - 3227 (2015/08/03)
Abstract A type of novel rhodanine-based 4-anilinoquinazoline, which designed the combination between quinazoline as the backbone and various substituted biological rhodanine groups as the side chain, have been synthesized, and their antiproliferative act