82703-35-3Relevant academic research and scientific papers
4-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)-3,6-DIHYDROPYRIDINE-1-(2H)-CARBOXAMIDE DERIVATIVES AS LIMK AND/OR ROCK KINASES INHIBITORS FOR USE IN THE TREATMENT OF CANCER
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Paragraph 0105; 0195; 0197, (2021/12/07)
The present invention concerns a compound of formula (I), in particular as LIMK and/or ROCK kinases inhibitors. The present invention also concerns these new inhibitors for use for the treatment of a condition selected in the group consisting of: cancers, virion infections, ocular hypertension and glaucoma formation, Neurofibromatosis type 1 and 2, psoriatic lesions, inflammatory diseases and hyperalgesia, central sensitization and chronic pain, reproduction erectile dysfunction, and neuronal diseases. The present description discloses the syntheses and characterisation of exemplary compounds as well as pharmacological data thereof (e.g. pages 32 to 127; examples 1 to 96; families 1 to 8; compounds; biological studies; tables). An exemplary compound is e.g. 4-(5-m ethyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-N-phenyl-3,6-dihydropyridine-1-(2H)-carboxamide (example 1; compound 5).
Synthesis of 7-Unsubstituted 7H-Pyrrolopyrimidines
Pichler, Herbert,Folkers, Gerd,Roth, Hermann J.,Eger, Kurt
, p. 1485 - 1505 (2007/10/02)
The title compounds 4 are obtained by N-7 dealkylation of the 2-furanylmethyl, 2-thiophenylmethyl, or 1-phenylethyl group from 2a-g and 10 a-j with polyphosphoric acid.In contrast to the 2-furanylmethyl group the 2-thiophenylmethyl and 1-phenylethyl group
