83784-81-0Relevant articles and documents
Chemoselective N-acylation of indoles and oxazolidinones with carbonylazoles
Heller, Stephen T.,Schultz, Erica E.,Sarpong, Richmond
supporting information; experimental part, p. 8304 - 8308 (2012/09/08)
Unique reactivity: In the presence of more reactive amine and alcohol functional groups and of carboxylic acids, the chemoselective N-acylation of indoles (see scheme) and oxazolidinones is achieved by taking advantage of the unique reactivity of carbonylazole acylating agents with catalytic amounts of 1,8-diazabicyclo[5.4.0]undec-7-ene (DBU). Copyright