847026-36-2Relevant academic research and scientific papers
N-Oxide analogs of WAY-100635: New high affinity 5-HT1A receptor antagonists
Marchais-Oberwinkler, Sandrine,Nowicki, Bartek,Pike, Victor W.,Halldin, Christer,Sandell, Johan,Chou, Yuan-Hwa,Gulyas, Balazs,Brennum, Lise T.,Farde, Lars,Wikstr?m, H?kan V.
, p. 883 - 893 (2007/10/03)
WAY-100635 [N-(2-(1-(4-(2-methoxyphenyl)piperazinyl)ethyl))-N-(2-pyridinyl) cyclohexanecarboxamide] 1 and its O-desmethyl derivative DWAY 2 are well-known high affinity 5-HT1A receptor antagonists, which when labeled with carbon-11 (β+/su
