866004-34-4Relevant academic research and scientific papers
11-(Pyridinylphenyl)steroids-A new class of mixed-profile progesterone agonists/antagonists
Rewinkel, Jos,Enthoven, Mark,Golstein, Irene,van der Rijst, Marcel,Scholten, Andre,van Tilborg, Martin,de Weys, Dirk,Wisse, Jeffry,Hamersma, Hans
, p. 2753 - 2763 (2008)
Recently, a new class (often referred to as SPRMs: selective progesterone receptor modulators) of progesterone receptor ligands with mixed agonist/antagonist properties has been described. Such compounds are envisaged, for example, as treatment for endome
PROGESTERONE RECEPTOR MODULATORS
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Page/Page column 20-21, (2010/02/14)
The subject invention provides a compound according to Formula I, wherein Formula (1) is O, NOH, NO(1-4C)alkyl, NO(1-4C)acyl; Al-A5 are C, substituted with RI, or N, provided that at least one and not more than three of Al-A5 are N; or one or two of Al, A
