869852-75-5Relevant academic research and scientific papers
Estrogen receptor β selective ligands: Discovery and SAR of novel heterocyclic ligands
Chesworth, Richard,Wessel, Matthew D.,Heyden, Lisa,Mangano, F. Michael,Zawistoski, Michael,Gegnas, Laura,Galluzzo, David,Lefker, Bruce,Cameron, Kimberly O.,Tickner, Jeanne,Lu, Bihong,Castleberry, Tessa A.,Petersen, Donna N.,Brault, Amy,Perry, Pia,Ng, Oicheng,Owen, Thomas A.,Pan, Lydia,Ke, Hua-Zhu,Brown, Thomas A.,Thompson, David D.,DaSilva-Jardine, Paul
, p. 5562 - 5566 (2007/10/03)
A series of ligands with varying heterocyclic cores and substituents that display a range of selectivity's (up to >100x) for ER-β over ER-α are reported.
