869959-33-1

Upstream product

• 15761-38-3 L-N-Boc-Ala 
• 10269-01-9 3-bromobenzylamine 

Downstream Products

• 916992-52-4 (1-{1-[1-(3-bromobenzylcarbamoyl)ethylcarbamoyl]-2-methylpropylcarbamoyl}-2-phenylethyl)carbamic acid tert-butyl ester 
• 916992-53-5 3-Amino-N-((S)-1-{(S)-1-[(S)-1-(3-bromo-benzylcarbamoyl)-ethylcarbamoyl]-2-methyl-propylcarbamoyl}-2-phenyl-ethyl)-benzamide 

Relevant academic research and scientific papers

Synthesis of cyclic peptides constrained with biarylamine linkers using Buchwald-Hartwig C-N coupling

In this paper, we describe the synthesis of conformationally constrained cyclic peptides with biarylamine linkers for peptidomimetics using palladium-catalyzed intramolecular Buchwald-Hartwig C-N coupling. We have prepared a variety of di-, tri-, and tetr

Synthesis of conformationally constrained cyclic peptides using an intramolecular Sonogashira coupling

Small peptides having a 3-bromobenzyl group at the C-termini and n-alkynoyl group at the N-termini undergo a smooth copper-free intramolecular Sonogashira coupling reaction to afford the corresponding cyclic peptides in moderate yields. Scope and limitati