873072-60-7Relevant articles and documents
Scaffold oriented synthesis. Part 1: Design, preparation, and biological evaluation of thienopyrazoles as kinase inhibitors
Akritopoulou-Zanze, Irini,Darczak, Daria,Sarris, Kathy,Phelan, Kathleen M.,Huth, Jeffrey R.,Song, Danying,Johnson, Eric F.,Jia, Yong,Djuric, Stevan W.
, p. 96 - 99 (2007/10/03)
We report the synthesis of kinase targeted libraries based on the thienopyrazole scaffold. Several thienopyrazole analogs have been identified as submicromolar inhibitors of KDR.