873446-68-5Relevant academic research and scientific papers
New fused benzazepine as selective D3 receptor antagonists. Synthesis and biological evaluation. Part 2: [g]-Fused and hetero-fused systems
Micheli, Fabrizio,Bonanomi, Giorgio,Braggio, Simone,Capelli, Anna Maria,Damiani, Federica,Di Fabio, Romano,Donati, Daniele,Gentile, Gabriella,Hamprecht, Dieter,Perini, Ornella,Petrone, Marcella,Tedesco, Giovanna,Terreni, Silvia,Worby, Angela,Heidbreder, Christian
, p. 908 - 912 (2008)
The synthesis and the SAR of a new series of potent and selective dopamine D3 receptor antagonists is reported. The new scaffolds of the [g]-fused and the hetero-fused tricyclic benzazepine are here reported together with their pharmacokinetic profile.
