874739-16-9Relevant academic research and scientific papers
An efficient desulfitative C-C cross coupling of fused thiazolidine-2-thione with boronic acids and boronic acid pinacol esters: Formation of fused thiazoles
Rajaguru, Kandasamy,Mariappan, Arumugam,Manjusri, Ramachandran,Muthusubramanian, Shanmugam,Bhuvanesh, Nattamai
, p. 86832 - 86839 (2015/11/03)
An efficient Pd(0)-catalyzed Cu(i)-mediated desulfitative C-C cross-coupling of benzo-fused thiazolidine-2-thione with boronic acids under neutral Liebeskind-Srogl conditions is described. The desulfitative cross coupling of boronic acid pinacol esters has also been demonstrated with fused thiazolidine-2-thione under basic conditions to afford fused thiazoles with good to excellent yields.
Solid phase combinatorial synthesis of benzothiazoles and evaluation of topoisomerase II inhibitory activity
Choi, Suk-June,Park, Hyen Joo,Lee, Sang Kook,Kim, Sang Woong,Han, Gyoonhee,Choo, Hea-Young Park
, p. 1229 - 1235 (2007/10/03)
To investigate one possible mechanism of action of the cytotoxic activity of benzothiazoles, we synthesized 2-(substituted-phenyl)benzothiazoles and evaluated their ability to inhibit topoisomerase II activities. Solid phase combinatorial method using tri
