874900-01-3Relevant articles and documents
THIAZOLE DERIVATIVES HAVING VAP-1 INHIBITORY ACTIVITY
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Page/Page column 83, (2008/06/13)
A compound of the formula (I), (II), (III) or (IV): wherein each symbol is as defined in the specification,or a pharmaceutically acceptable salt thereof useful as a vascular adhesion protein-1 (VAP-1) inhibitor, a pharmaceutical composition, a method for preventing or treating a VAP-1 associated disease, especially macular edema, which method includes administering an effective amount of the compound or a pharmaceutically acceptable salt thereof to a subject, and the like.
THIAZOLE DERIVATIVES AND THEIR USE AS VAP-1 INHIBITORS
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Page 116-117, (2010/02/07)
A compound of the formula (I): R1-NH-X-Y-Z (I) wherein R1 is acyl; X is a bivalent residue derived from optionally substituted thiazole; Y is a bond, lower alkylene or -COHN-; and Z is a groupe of the formulae (II) or (III) wherein R