879553-92-1Relevant articles and documents
Fragment-based drug design targeting syntenin PDZ2 domain involved in exosomal release and tumour spread
Garcia, Manon,Hoffer, Laurent,Leblanc, Rapha?l,Benmansour, Fatiha,Feracci, Mikael,Derviaux, Carine,Egea-Jimenez, Antonio Luis,Roche, Philippe,Zimmermann, Pascale,Morelli, Xavier,Barral, Karine
, (2021/07/09)
Syntenin stimulates exosome production and its expression is upregulated in many cancers and implicated in the spread of metastatic tumor. These effects are supported by syntenin PDZ domains interacting with syndecans. We therefore aimed to develop, throu