88012-49-1Relevant academic research and scientific papers
Nucleophilic substitution of azide acting as a pseudo leaving group: One-step synthesis of various aza heterocycles
Doebelin, Christelle,Schmitt, Martine,Antheaume, Cyril,Bourguignon, Jean-Jacques,Bihel, Frederic
, p. 11335 - 11341 (2013)
The reaction of 3-azidopropanoic acid with the carbodiimide-based coupling reagent DIC leads to a six-membered-ring intermediate acting as a versatile precursor to a diverse set of aza heterocycles, including mono-, bi-, and tricyclic compounds.
Neuroleptic 3-azetidinylethyl-1-phenyl-2-imidazolidinones
-
, (2008/06/13)
New 3-azetidinylethyl-1-phenyl-2-imidazolidinones with neuroleptic activity, their use and methods for their preparation. The azetidinyl group bears alkyl substituents in position 3 and the phenyl group bears halogenated substituents in position 3 and hydroxy group or acylated hydroxy groups in position 4 and/or 6.
