889673-71-6Relevant articles and documents
2,6-Disubstituted and 2,6,8-trisubstituted purines as adenosine receptor antagonists
Chang, Lisa C. W.,Spanjersberg, Ronald F.,Von Frijtag Drabbe Künzel, Jacobien K.,Mulder-Krieger, Thea,Brussee, Johannes,Ijzerman, Adriaan P.
, p. 2861 - 2867 (2007/10/03)
Purines have long been exploited as adenosine receptor antagonists. The substitution pattern about the purine ring has been well investigated, and certain criteria have become almost a prerequisite for good affinity at the adenosine A1 receptor