89060-59-3Relevant academic research and scientific papers
Design, synthesis and biological evaluation of glycolamide, glycinamide, and β-amino carbonyl 1,2,4-triazole derivatives as DPP-4 inhibitors
Fuh, Mao-Tsu,Tseng, Ching-Chun,Li, Sin-Min,Tsai, Shuo-En,Chuang, Tsung-Jui,Lu, Chih-Hao,Yang, Ya-Chen,Tsai, Henry J.,Wong, Fung Fuh
supporting information, (2021/06/21)
Through modification of the skeleton of Sitagliptin and Vildagliptin, we successfully synthesized and built-up four series of 1,2,4-triazole derivatives, containing N,O-disubstituted glycolamide, N,N′-disubstituted glycinamide, β-amino ester, and β-amino
