893386-19-1Relevant academic research and scientific papers
THIENO-PYRIDINE DERIVATIVES AS GABA-B ALLOSTERIC ENHANCERS
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Page/Page column 34, (2008/06/13)
The present invention relates to compounds of formula (I), Wherein R1 to R5 are as defined in the specification which compounds are active on the GABABreceptor and can be used for the manufacture of medicaments useful for treating CNS disorders.
Microwave-assisted synthesis of thieno[2,3-c]pyridine derivatives as a new series of allosteric enhancers at the adenosine A1 receptor
Romagnoli, Romeo,Baraldi, Pier Giovanni,Moorman, Allan R.,Iaconinoto, Maria Antonietta,Carrion, Maria Dora,Cara, Carlota Lopez,Tabrizi, Mojgan Aghazadeh,Preti, Delia,Fruttarolo, Francesca,Baker, Stephen P.,Varani, Katia,Borea, Pier Andrea
, p. 5530 - 5533 (2007/10/03)
The microwave-assisted aromatization method has been used for the synthesis of a series of novel thieno[2,3-c]pyridines. This rapid method produces compounds in good yield within minutes in comparison with conventional heating method. The synthesized mole
