895524-76-2Relevant academic research and scientific papers
Optimization of pyrazole inhibitors of Coactivator Associated Arginine Methyltransferase 1 (CARM1)
Huynh, Tram,Chen, Zhong,Pang, Suhong,Geng, Jieping,Bandiera, Tiziano,Bindi, Simona,Vianello, Paola,Roletto, Fulvia,Thieffine, Sandrine,Galvani, Arturo,Vaccaro, Wayne,Poss, Michael A.,Trainor, George L.,Lorenzi, Matthew V.,Gottardis, Marco,Jayaraman, Lata,Purandare, Ashok V.
scheme or table, p. 2924 - 2927 (2010/03/03)
Design, synthesis, and SAR development led to the identification of the potent, novel, and selective pyrazole based inhibitor (7f) of Coactivator Associated Arginine Methyltransferase (CARM1).
Inhibitors of protein arginine methyl transferases
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Page/Page column 83, (2010/11/26)
A compound of formula I, or a stereoisomer, a tautomer, a pharmaceutically acceptable salt or solvate thereof, methods of using such compounds in the treatment of hyperproliferative, inflammatory, infectious, and immunoregulatory disorders and diseases; a
