898252-79-4Relevant articles and documents
Discovery of indole-containing tetracycles as a new scaffold for androgen receptor ligands
Zhang, Xuqing,Li, Xiaojie,Allan, George F.,Musto, Amy,Lundeen, Scott G.,Sui, Zhihua
, p. 3233 - 3237 (2006)
A novel series of tetracyclic indoles have been designed, synthesized and evaluated as androgen receptor (AR) ligands. Studies of structure-activity relationships (SARs) were investigated, which led to some compounds in this series as strong binders to an