900019-83-2Relevant academic research and scientific papers
INHIBITORS OF VAP-1
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Paragraph 0338-0339; 0400; 0520, (2020/05/12)
Provided herein are compounds and methods of use thereof for the modulation of VAP-1 activity.
Diastereo- and enantioselective Pd(II)-catalyzed additions of 2-alkylazaarenes to N -boc imines and nitroalkenes
Best, Daniel,Kujawa, Szymon,Lam, Hon Wai
supporting information, p. 18193 - 18196 (2013/01/15)
A chiral Pd(II)-bis(oxazoline) complex was found to be highly effective in promoting the first direct diastereo- and enantioselective addition of alkylazaarenes to N-Boc aldimines and nitroalkenes under mild conditions. Deprotection of Boc-protected products proceeded readily to provide amines in high yields.
