905752-13-8

Upstream product

• 155020-44-3 2-fluoro-1,3-dimethoxy-4-nitrobenzene 
• 771-69-7 2,3,4-trifluoronitrobenzene 
• 195136-66-4 1-amino-3-fluoro-2,4-dimethoxybenzene 

Downstream Products

• 1401998-80-8 3-fluoro-2,4-dihydroxybenzaldehyde 
• 502483-90-1 3-fluoro-2,4-dimethoxybenzaldehyde 
• 905752-14-9 4-(2,4-dimethoxy-3-fluoro-phenylethynyl)-1-methyl-1H-pyrazole 

Relevant academic research and scientific papers

1 -HYDROXY-BENZOOXABOROLES AS ANTIPARASITIC AGENTS

Provided are compounds useful for controlling endoparasites both in animals and agriculture. Further provided are methods for controlling endoparasite infestations of an animal by administering an effective amount of a compound as described above, or a pharmaceutically acceptable salt thereof, to an animal, as well as formulations for controlling endoparasite infestations using the compounds described above or an acceptable salt thereof, and an acceptable carrier. The claimed compounds are described by the following Markush formula:A typical example for a compound according to above formula is: A typical example for a compound according to above formula is:

CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS

The present invention relates to compounds of formula (I) for treating diseases associated with cysteine protease activity. The compounds are reversible inhibitors of cysteine proteases, including cathepsins B, K, C, F, H, L, O, S, W and X. Of particular interest are diseases associated with Cathepsin K.

NOVEL TUBULIN POLYMERISATION INHIBITORS

The present invention relates to compounds of general formula (I) as tublin polymerisation inhibitors and methods for preparing such compounds.