911292-61-0Relevant academic research and scientific papers
Synthesis of alkylated sugar amino acids: Conformationally restricted l-Xaa-l-Ser/Thr mimics
Risseeuw, Martijn D.P.,Mazurek, Jaroslaw,Van Langenvelde, Arjan,Van Der Marel, Gijsbert A.,Overkleeft, Herman S.,Overhand, Mark
, p. 2311 - 2314 (2008/02/14)
Two synthetic strategies for the generation of δ-substituted pyranoid sugar amino acids (SAAs) are evaluated. The first employs chiral nonracemic tert-butane sulfinamides as key reagents. Regardless of the stereochemistry of the applied sulfinamide, the p
Stereoselective one-pot synthesis of constrained N,O-orthogonally protected C-glycosyl norstatines [C(1′)-aminoglycosyl-1,3-dioxolan-4-ones]
Guerrini, Andrea,Varchi, Greta,Battaglia, Arturo
, p. 6785 - 6795 (2007/10/03)
A procedure for the synthesis of conformationally constrained C-glycosyl norstatines has been developed. The key step of the reaction is the addition of (S)-N-sulfinyl azomethines to chiral (2S)-enolates of dioxolanones which exploits Seebach's "SRS" prin
