91533-09-4

Upstream product

• 619-17-0 4-Nitroanthranilic acid 

Downstream Products

• 129175-53-7 (S)-2-[4-[(2-Methyl-4-oxo-3,4-dihydro-quinazolin-6-ylmethyl)-prop-2-ynyl-amino]-2-(2,2,2-trifluoro-acetylamino)-benzoylamino]-pentanedioic acid diethyl ester 
• 129175-55-9 (S)-2-[4-[Ethyl-(2-methyl-4-oxo-3,4-dihydro-quinazolin-6-ylmethyl)-amino]-2-(2,2,2-trifluoro-acetylamino)-benzoylamino]-pentanedioic acid diethyl ester 
• 129175-54-8 (S)-2-[4-[Methyl-(2-methyl-4-oxo-3,4-dihydro-quinazolin-6-ylmethyl)-amino]-2-(2,2,2-trifluoro-acetylamino)-benzoylamino]-pentanedioic acid diethyl ester 
• 129193-64-2 (S)-2-{2-Amino-4-[(2-methyl-4-oxo-3,4-dihydro-quinazolin-6-ylmethyl)-prop-2-ynyl-amino]-benzoylamino}-pentanedioic acid 
• 129175-34-4 (S)-2-{2-Amino-4-[ethyl-(2-methyl-4-oxo-3,4-dihydro-quinazolin-6-ylmethyl)-amino]-benzoylamino}-pentanedioic acid 
• 129175-33-3 (S)-2-{2-Amino-4-[methyl-(2-methyl-4-oxo-3,4-dihydro-quinazolin-6-ylmethyl)-amino]-benzoylamino}-pentanedioic acid 
• 129175-77-5 (S)-2-[4-Prop-2-ynylamino-2-(2,2,2-trifluoro-acetylamino)-benzoylamino]-pentanedioic acid diethyl ester 
• 129175-84-4 (S)-2-[4-Nitro-2-(2,2,2-trifluoro-acetylamino)-benzoylamino]-pentanedioic acid diethyl ester 
• 129175-79-7 (S)-2-[4-Ethylamino-2-(2,2,2-trifluoro-acetylamino)-benzoylamino]-pentanedioic acid diethyl ester 
• 129175-78-6 (S)-2-[4-Methylamino-2-(2,2,2-trifluoro-acetylamino)-benzoylamino]-pentanedioic acid diethyl ester 
• 129175-80-0 (S)-2-[4-Amino-2-(2,2,2-trifluoro-acetylamino)-benzoylamino]-pentanedioic acid diethyl ester 

Relevant academic research and scientific papers

Benzyl-piperidine derivatives

Benzly-piperidine derivatives of formula I and their pharmaceutically acceptable salts are used in the control of psychotic disorders which are caused by damage to the dopamine system, especially schizophrenia. STR1 A is STR2 B is STR3 R 1, R 2 and R 3 are independently hydrogen, amino, nitro, halogen, lower-alkly or lower-alkoxy. R 4, R 5 and R 6 are independently hydrogen, nitro, halogen, lower-alkyl, lower-alkoxy, cyano, trifluoromethyl, amino, lower-alkylamino or di-lower-alkylamino. R 7, R 2 and R 9 are independently hydrogen, amino or nitro.

Fungicidal acylamidobenzamides

Fungicidal compounds having the formula (I): in which D and E are independently H or F; X and Y are 0 or S; R1 to R4 have various specified values; A and B are independently H, iodo, nitro, cyano, C1 4 alkoxycarbonyl, Csu

4H-3,1-BENZOXAZIN-4-ONE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE INHIBITION OF SERINE PROTEASES

A 4H-3,1-benzoxazin-4-one compound of the formula (I): STR1 wherein R is a hydrogen atom or alkyl radical, A is an amino acid residue or a peptide having 2 to 3 amino acid residues, which amino acid residue may have a side chain thereof protected by a protective radical, X is an alkyl, fluoroalkyl, OR 1 or NHR 1 radical wherein R 1 is an alkyl radical, and Y is a protective radical for an amino radical, and salts thereof, exhibit an excellent inhibitory activity against serine proteases, especially against human leukocyte elastase, and thus are useful as an effective component of a medicine for inhibiting elastase.