915409-65-3Relevant academic research and scientific papers
Tricyclic HIV integrase inhibitors V. SAR studies on the benzyl moiety
Jin, Haolun,Metobo, Sammy,Jabri, Salman,Mish, Michael,Lansdown, Rachael,Chen, Xiaowu,Tsiang, Manuel,Wright, Matthew,Kim, Choung U.
scheme or table, p. 2263 - 2265 (2009/12/07)
SAR studies on the para-fluorobenzyl moiety of tricyclic HIV integrase inhibitors are discussed and lead compounds with potency and PK properties comparable to raltegravir were identified.
Integrase inhibitor compounds
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Page/Page column 111-112, (2010/11/26)
Tricyclic compounds, protected intermediates thereof, and methods for inhibition of HIV-integrase are disclosed.
