915714-94-2

Downstream Products

• 915713-07-4 (S)-4-methylnaphthalene-1-sulfonic acid (3-amino-1-benzyl-oxymethylpropyl)amide 
• 915713-08-5 (S)-4-methylnaphthalene-1-sulfonic acid (1-benzyloxymethyl-3-guanidinylpropyl)amide 
• 915714-25-9 (S)-4-methylnaphthalene-1-sulfonic acid [1-benzyloxymethyl-3-(N,N'-bis(Boc)guanidinyl)propyl]amide 

Relevant academic research and scientific papers

PEPTIDOMIMETICS SELECTIVE FOR THE SOMATOSTATIN RECEPTOR SUBTYPES 1 AND/OR 4

The invention relates to (hetero)arylsulfonylamino based peptidomimetics of formula (I), wherein A, D, E, J, Q1 R1 , R2, R3, p and j are defined as disclosed, or a pharmaceutically acceptable salt or ester thereof. Compounds of formula (I) possess high affinity and selectivity for the somatostatin receptor subtypes sst1 and/or sst4 and can be used for the treatment or diagnosis of diseases or conditions wherein sst1 and/or sst4 agonists or antagonists are indicated to be useful.