923253-36-5Relevant articles and documents
Copper-catalyzed direct oxidation and N-arylation of benzylamines with diaryliodonium salts
Liu, Xin,Mao, Dan,Wu, Shengying,Yu, Jianjun,Hong, Gang,Zhao, Qiao,Wang, Limin
, p. 1132 - 1136 (2014)
An efficient approach for the synthesis of N-arylated amides was developed via copper(II) triflate-catalyzed direct oxidation of (aryl)methylamines to primary arylamides by air and subsequent N-arylation by diaryliodonium salts. Various substituted benzylamines could be applied in the reaction, providing a series of N-arylated amides in moderate to good yields. This method showed convenient, practical, and environment friendly advantages.