928658-24-6Relevant articles and documents
Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands
Salama, Ismail,Hocke, Carsten,Utz, Wolfgang,Prante, Olaf,Boeckler, Frank,Hübner, Harald,Kuwert, Torsten,Gmeiner, Peter
, p. 489 - 500 (2007)
Elucidation of the physiological role of the D3 receptor and its distribution in the brain using positron emission tomography (PET) is hampered by the lack of bioavailable subtype selective tracer ligands. To develop appropriate D3 r
AZETIDINYL G-PROTEIN COUPLED RECEPTOR AGONISTS
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Page/Page column 22, (2009/05/28)
Compounds of formula (I): or pharmaceutically acceptable salts thereof, are agonists of GPR119 and are useful for the treatment of diabetes and as peripheral regulators of satiety, e.g. for the treatment of obesity and metabolic syndrome.