933020-73-6Relevant articles and documents
Simple strategy for sulfonyl ethynylogs of coumarins
Guravaiah, Nalajam,Rao, Vedula Rajeswar
, p. 2693 - 2700 (2011)
Synthesis of 3-(2-(phenylsulfonyl) ethynyl)-2H-chromen-2-one is described. Reaction of β-ketosulfones with semicarbazide hydrochloride in ethanol at reflux temperature gave the corresponding semicarbazones, which on oxidative cyclization with selenium dioxide resulted in the formation of the corresponding 1,2,3-selenodiazole derivatives. These on pyrolysis gave the titled compounds. Taylor & Francis Group, LLC.
Novel 3-substituted coumarins as selective human carbonic anhydrase IX and XII inhibitors: Synthesis, biological and molecular dynamics analysis
Abdelrahman, Mohamed A.,Ibrahim, Hany S.,Nocentini, Alessio,Eldehna, Wagdy M.,Bonardi, Alessandro,Abdel-Aziz, Hatem A.,Gratteri, Paola,Abou-Seri, Sahar M.,Supuran, Claudiu T.
, (2020/10/09)
In this study, diverse series of coumarin derivatives were developed as potential carbonic anhydrase inhibitors (CAIs). A “tail” approach was adopted by selecting the coumarin motif as a tail that is connected to the ZBG benzenesulfonamide moiety via a hy
Synthesis of a new class of Sulfone-linked 3-([1,2,3]-thiadazol-4-yl)- chromen-2-ones
Guravaiah, Nalajam,Rao, Vedula Rajeswar
scheme or table, p. 361 - 367 (2010/06/19)
A new class of 3-[5-(phenylsulfonyl)1,2,3-thiadizol-4-yl)-2H-chromen-2-ones (5) has been prepared from 3-(2-(phenylsulfonyl)-2H-chromen-2-ones (4).
Solvent-free synthesis of new heteryl β-ketosulfones
Guravaiah, Nalajam,Rao, Vedula Rajeswar
experimental part, p. 87 - 89 (2009/11/30)
A novel efficient method for the coupling of sulfinic acid salts and α-halo ketones is described. A variety of heteryl β-ketosulfones have been formed in an excellent yields at room temperature under solvent-free conditions.