934542-72-0Relevant articles and documents
Integrated cross-coupling strategy for an -carboline-based aurora b kinase inhibitor
Mineno, Masahiro,Sera, Misayo,Ueda, Tsuyoshi,Mizufune, Hideya,Zanka, Atsuhiko,Obryan, Colin,Brown, Jason,Scorah, Nick
, p. 1564 - 1568 (2015/02/19)
An efficient and practical synthetic process for an α-carboline-based Aurora B kinase inhibitor was achieved using an integrated Pd-catalyzed cross-coupling strategy. The process features a mild and efficient method for construction of the α-carboline cor
POLYMORPHS OF 5-(3-(ETHYLSULFONYL)PHENYL)-3,8-DIMETHYL-N-(1-METHYLPIPERIDIN-4-YL)-9H-PYRIDO[2,3-B]INDOLE-7-CARBOXAMIDE AND METHODS OF USE THEREFOR
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Page/Page column 48-49, (2009/12/02)
The invention relates to polymorphic forms of 5-(3-(ethylsulfonyl)phenyl)-3,8-dimethyl-N-(1-methylpiperidin-4-yl)-9h-pyrido[2,3-b]indole-7-carboxamide (referred to herein as Compound I), which has the formula: (A). The invention also relates to compositio
KINASE INHIBITORS
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Page/Page column 174-175, (2010/11/27)
Compounds, pharmaceutical compositions, kits and methods are provided for use with kinases that comprise a compound selected from the group consisting of formula (I) wherein the variables are as defined herein.