935472-63-2Relevant academic research and scientific papers
An approach to?the?stereo-controlled synthesis of?polycyclic derivatives of?l-4-thiazolidinecarboxylic acid active against?HIV-1?integrase
Aiello,Brizzi,De Grazia,Garofalo,Grande,Sinicropi,Dayam,Neamati
, p. 914 - 917 (2007/10/03)
Herein, we describe a new strategy for the preparation of thiazolothiazepine-based inhibitors of human immunodeficiency virus type-1 integrase (IN). The present method allows facile preparation of the title compounds in a single enantiomeric form starting
