938186-08-4Relevant academic research and scientific papers
Novel selective human melanocortin-3 receptor ligands: Use of the 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one (Aba) scaffold
Ballet, Steven,Mayorov, Alexander V.,Cai, Minying,Tymecka, Dagmara,Chandler, Kevin B.,Palmer, Erin S.,Rompaey, Karolien Van,Misicka, Aleksandra,Tourwe, Dirk,Hruby, Victor J.
, p. 2492 - 2498 (2008/02/02)
In search of new selective antagonists and/or agonists for the human melanocortin receptor subtypes hMC1R to hMC5R to elucidate the specific biological roles of each GPCR, we modified the structures of the superagonist MT-II (Ac-Nle-c[Asp-His-d-Phe-Arg-Tr
