93826-89-2Relevant articles and documents
Cu-Mediated Radiofluorination of Aryl Pinacolboronate Esters: Alcohols as Solvents with Application to 6-L-[18F]FDOPA Synthesis
Fedorova, Olga,Krasikova, Raisa,Kuznetsova, Olga,Orlovskaya, Viktoriya
, p. 7079 - 7086 (2020)
Cu-mediated radiofluorination of arylboronic acid pinacol esters (ArylBPin) using Cu(OTf)2(Py)4 complex is a useful approach for the introduction of [18F]fluorine into non-activated arenes and heteroarenes. Owing to the co
MCR scaffolds get hotter with 18F-Labeling
Zarganes-Tzitzikas, Tryfon,Clemente, Gon?alo S.,Elsinga, Philip H.,D?mling, Alexander
, (2019/04/16)
Imaging techniques, such as positron emission tomography (PET), represent great progress in the clinical development of drugs and diagnostics. However, the efficient and timely synthesis of appropriately labeled compounds is a largely unsolved problem. Nu
An azeotropic drying-free approach for copper-mediated radiofluorination without addition of base
Zhang, Xiang,Basuli, Falguni,Swenson, Rolf E.
, p. 139 - 145 (2019/02/25)
Copper-mediated radiofluorination provides a quick and versatile approach for 18F-labeling of arenes and heteroarenes. However, this method is known to be base sensitive, which has been a barrier for preparative scale radiosynthesis. In this re