93988-49-9Relevant academic research and scientific papers
Identification of benzothiophene amides as potent inhibitors of human nicotinamide phosphoribosyltransferase
Chen, Wei,Dong, Guoqiang,He, Shipeng,Xu, Tianying,Wang, Xia,Liu, Na,Zhang, Wannian,Miao, Chaoyu,Sheng, Chunquan
, p. 765 - 768 (2016)
Nicotinamide phosphoribosyltransferase (Nampt) is an attractive therapeutic target for cancer. A Nampt inhibitor with novel benzothiophene scaffold was discovered by high throughput screening. Herein the structure-activity relationship of the benzothiophe
