940950-96-9Relevant academic research and scientific papers
Unified azoline and azole syntheses by optimized aza-wittig chemistry
Loos, Patrick,Ronco, Cyril,Riedrich, Matthias,Arndt, Hans-Dieter
supporting information, p. 3290 - 3315 (2013/06/27)
Intramolecular aza-Wittig ring closures were applied to synthesize thiazolines, oxazolines, and imidazolines from β-azido thioester, ester, and amide precursors. The cyclization precursors were obtained from amino acid derivatives. Optimized conditions fo
Peptide-embedded heterocycles by mild single and multiple aza-Wittig ring closures
Riedrich, Matthias,Harkal, Surendra,Arndt, Hans-Dieter
, p. 2701 - 2703 (2008/02/14)
Ring a ring o'azoles: The aza-Wittig cyclization of amino acids and peptides is extremely mild, selective, and versatile. The reaction of amino acid esters and amino acid thioester azides delivers peptidic 1,3-azolines and 1,3-azoles with unsurpassed func
